Design, synthesis and evaluation of (E)-1-(4-(2-(1H-pyrazol-5-yl)vinyl)phenyl) derivatives as next generation selective RET inhibitors overcoming RET solvent front mutations (G810C/R)

• DOI: 10.1016/j.ejmech.2025.117294
• Publication Date: 2025-01-24T00:05:24Z
• Authors: Mingjin Xu; Kaifu Wu; Rui He; Jiahuan He; Gangpeng Yang; Haowen Ma; Lijie Peng; Shuyao Zhang; Li Tan; Zhang Zhang; Qian Cai