An Efficient Synthesis of N-Protected β-Aminoethanesulfonyl Chlorides: Versatile Building Blocks for the Synthesis of Oligopeptidosulfonamides

• DOI: 10.1055/s-2000-7615
• Publication Date: 2002-07-26T07:45:05Z
• Authors: Arwin J. Brouwer; Menno C. F. Monnee; Rob M. J. Liskamp
• Keywords: Sulfonyl

A very efficient method for the synthesis of β-aminoethanesulfonyl chlorides is described. These aliphatic functionalized sulfonyl are accessible starting from a variety protected amino acids, including those having side chains.