Joan Jair Espinoza-Rodríguez

ORCID: 0009-0000-7413-0826
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About
Contact & Profiles
Research Areas
  • Cancer therapeutics and mechanisms
  • Antibiotic Resistance in Bacteria
  • Antibiotics Pharmacokinetics and Efficacy

Universidad Autónoma de Zacatecas "Francisco García Salinas"
2023

Structure–activity relationship (SAR) studies allow the evaluation of between structural chemical changes and biological activity. Fluoroquinolones have characteristics that their structure to be modified new analogs with different therapeutic properties generated. The objective this research is identify select C-7 heterocycle fluoroquinolone analog (FQH 1–5) antibacterial activity similar reference through in vitro, silico, vivo evaluations. First, SAR analysis was conducted on FQH 1–5,...

10.3390/molecules28166018 article EN cc-by Molecules 2023-08-11
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